Compile Data Set for Download or QSAR
maximum 50k data
Found 28 of ic50 data for polymerid = 49000978
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50240455(CHEMBL1253351)
Affinity DataIC50:  0.280nMAssay Description:Antagonist activity at rat P2X1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50540410(CHEMBL337395)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at rat P2X1 receptorMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102298(4-(4-Formyl-5-hydroxy-6-methyl-3-phosphonomethyl-p...)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102295(4-(4-Formyl-5-hydroxy-6-methyl-3-phosphonooxymethy...)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102299(2-(4-Formyl-5-hydroxy-6-methyl-3-phosphonomethyl-p...)
Affinity DataIC50:  11nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102300(CHEMBL331250 | [4-(4-Formyl-5-hydroxy-6-methyl-3-p...)
Affinity DataIC50:  12nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50118221(9H-purine derivative | CHEMBL132722 | DIPHOSPHOMET...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102301(4-[4-Formyl-5-hydroxy-6-methyl-3-(2-phosphono-ethy...)
Affinity DataIC50:  20nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102296(2-(4-Formyl-5-hydroxy-6-methyl-3-phosphonomethyl-p...)
Affinity DataIC50:  37nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102304(CHEMBL116926 | Phosphoric acid mono-(4-formyl-5-hy...)
Affinity DataIC50:  42nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102297(CHEMBL118007 | [2-(3,5-Bis-phosphonomethyl-phenyla...)
Affinity DataIC50:  42nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50102295(4-(4-Formyl-5-hydroxy-6-methyl-3-phosphonooxymethy...)
Affinity DataIC50:  43nMAssay Description:Antagonist activity at recombinant rat P2X1 receptor expressed in Xenopus oocytes assessed as ion flux stimulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50064800(2-(4-Formyl-5-hydroxy-6-methyl-3-phosphonooxymethy...)
Affinity DataIC50:  43nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM85043(CAS_149017-66-3 | CHEMBL69234 | NSC_6093163 | PPAD...)
Affinity DataIC50:  99nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336781(CHEMBL1672104 | Disodium 1-Amino-4-[3-(4,6-dichlor...)
Affinity DataIC50:  422nMAssay Description:Antagonist activity against rat P2X1 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50540409(CHEBI:34941 | CHEMBL69234)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat P2X1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat P2X1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50118245(CHEMBL133572 | MG 40-3)
Affinity DataIC50:  1.60E+3nMAssay Description:The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) like receptor from rat vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50168286(1H-Benzoimidazole-2-carboxylic acid [(R)-1-((1S,2R...)
Affinity DataIC50:  3.00E+3nMAssay Description:Antagonist activity at rat P2X1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataIC50:  4.68E+3nMAssay Description:Antagonist activity at P2X1 receptor in rat vas deferens assessed as inhibition of alpha/beta-meATP-induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50336781(CHEMBL1672104 | Disodium 1-Amino-4-[3-(4,6-dichlor...)
Affinity DataIC50:  4.70E+3nMAssay Description:Antagonist activity at P2X1 receptor in rat vas deferens assessed as inhibition of alphabeta me-ATP-induced responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50118237(CHEMBL130059 | Uniblue A)
Affinity DataIC50:  7.50E+3nMAssay Description:The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) from rat vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50118218(CHEMBL131271 | Disodium 1-amino-4-[4-(4,6-dichloro...)
Affinity DataIC50:  8.80E+3nMAssay Description:The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) like receptor from rat vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50118231(CHEMBL134193 | Cibachron Blue 3GA)
Affinity DataIC50:  9.60E+3nMAssay Description:The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) from rat vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50064801(2-(4,7-Dihydroxy-3-methyl-7-oxo-5,9-dihydro-6,8-di...)
Affinity DataIC50:  1.02E+4nMAssay Description:Compound was tested in a functional ion channel assay of ATP-induced current at recombinant rat P2X1 receptor expressed in Xenopus oocytes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50064801(2-(4,7-Dihydroxy-3-methyl-7-oxo-5,9-dihydro-6,8-di...)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of inward ion current elicited by ATP at P2X1 receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50064800(2-(4-Formyl-5-hydroxy-6-methyl-3-phosphonooxymethy...)
Affinity DataIC50:  4.25E+4nMAssay Description:Compound was tested in a functional ion channel assay of ATP-induced current at recombinant rat P2X1 receptor expressed in Xenopus oocytes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(RAT)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM85043(CAS_149017-66-3 | CHEMBL69234 | NSC_6093163 | PPAD...)
Affinity DataIC50:  9.85E+4nMAssay Description:Compound was tested in a functional ion channel assay of ATP-induced current at recombinant rat P2X1 receptor expressed in Xenopus oocytes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed